24.05.19 () 01:02

Dailypharm

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üADC ҰK-̿, R&D
2024-03-19 05:50:40
üADC ҰK-̿, R&D
2024-03-19 05:50:40

5Ϻ 10ϱ ̱ȸ мȸ(AACR 2024)

ѡѹ̡̺񿤹̿ ü 鿪׾ ĺ Ұ

, ADC ü ӻ

[ϸ= ] ı ӻ Ȥ ǥϰ ִ ̿ žĺ ۷ι 뿡 . ̿ ü, ü๰ü(ADC) ۷ι ֽ Ʈ带 ݿ žĺ ⿡ . Ѿ, ѹ̾ǰ, ̺񿤹̿, ͹̿ ӻ ϸ غ ƴ.

19 迡 ̱ȸ мȸ(AACR 2024) 5Ϻ 5ϰ ̱ ̰ ֵȴ. ̱ȸ ̱ӻȸ(ASCO), ȸ(ESMO) Բ 3 ȸ зǸ ӻ, ӻ1 ׾Ͻž ĺ ʱ ӻ ַ Ұȴ.

ΰ Ÿϴ ü, Ȱ

̹ AACR 2024 ű Ÿϴ ü ĺ ӻ ȴ. ü ϳ ̸ Ÿϴ Ŭü Ư ׿ ߰ ־ ӻ ٴ 򰡸 ް ִ.

Ѿ ̿ó 鿪׾ ü ӻ 2 Ѵ.

ȸ ʷ Ǵ žĺ YH41723̴. YH41723 Ѿ ̹ÿ½þư 鿪׾ PD-L1 TIGIT ŸѴ. Ѿ ŰƮ, ɵ ȭ 鿪׾ Ÿϴ PD-L1 鿪 T NK ǥ鿡 ϼ TIGIT(T-cell iMMunoreceptor with immunoglobulin and ITIM domain) Ÿ ȿ شȭϰڴٴ ȹ̴. Ѿ ܿ ν, ũ, Ƽ, 渮 ۷ι TIGIT Ÿϴ ׾ ž ϰ ִ.

̿ܿ Ѿ ̺񿤹̿ 鿪׾ YH32367 ӻ ͷ Ѵ. YH32367 ֿ Ͽ Ǵ ̿Ŀ HER2 41BB ܹ ŸѴ. PD-L1 ϴ ϼ ֺ 鿪 41BB ȰȭDZ 41BB ۿ ּȭϸ ׾ ȿ Ÿ ˷ ִ.

ѹ̾ǰ PD-L1 41BB Ÿϴ BH3120 ӻ ǥѴ. BH3120 ѹ̾ǰ ÷ Žٵ ƴ. ̴ 鿪 Ȱȭϴ ÿ Ÿ ϼ ϴ ü ÷ ̴. ̹ мȸ PD-1 뿡 ׾ ó ȿ Ͽ ̴. BH3120 ϰѹ̾ǰ ӻ ֵϰ ܵ ӻ1 ǰ ִ.

ѹ̾ǰ EZH1/2 HM97662 ǥѴ. EZH2 EZH1 Ȱȭ ߵǴ ˷ ִ. ѹ̾ǰ EZH1 EZH2 ϴ EZH2 ܵ غ ȿ ִٴ HM97662 ϰ ִ.

̺񿤹̿ ̹ мȸ ο ü 鿪׾ ABL112 ABL407 ӻ ͷ Ѵ. žĺ 9 AACR 2024 ǥ Ǵ ű ̴. ABL112 ABL407 41BB ü ÷ ׷ٵ-T ƴ. ABL112 TIGIT, ABL407 鿪 ϴ LILRB4 ǥѴ.

鿪 õ 鿪 ÿ ϴ ٵ ü ʸø ǥѴ. ȸ PD-L1 õ 鿪 CD47 ÿ ۿ ϼ 鿪ȸ ؿ ׾ȿ ̴. ʸø 󵵿 Ű ʾ CD47 ü ۿ Ÿ ʴ ˷ ִ.


͹̿, ADC ü LCB36 ӻ ù

ü๰ü(ADC) ϰ ִ ͹̿ ̹ мȸ ADC ü LCB36 ӻ ó Ѵ. LCB36 CD20 CD22 Ÿϴ ADC. CD20̳ CD22 Ÿϴ Ŭü CD20XCD3 Ÿϴ ü ߵ CD20 CD22 Ÿϴ LCB36 ʴ.

CD20 CD22 ׾Ͽ Ǵ ˷ ͹̿ LCB36 B Ÿϴ ž ϰ ִ. ͹̿ 콺 𵨿 ༺ ȹ̴.

̿ܿ ͹̿ Ŭ 18.2 ǥ ADC LCB02A ȹ̴. Ŭ 18.2 ַ ĵϿ Ǵ ܹ, ֱ ADC ž о߿ ޺λϴ ǥ̴.

͹̿ TROP2 ǥϴ ADC LCB84 ӻ Ѵ. LCB84 12 ̱ ص(J&J) ȸ Ἶ 17 ޷( 2 2400) Ը ⿡ žĺ̴.

ӻ󿡼 LCB84 ̼ҸӶ ̷ε TROP2 ADC ๰ ϴ Ͽ ȿ ִ. ̼ҸӶ (ƮƮָ轺ĭ) ֿ ADC ̴.

TROP2 Į ȣ ȯ İ Ѵ. ش ܹ ϳ ϼ ϴ ๰׼ ִ ˷.

TROP2 ̿Ŀ ַ , Ҽ,  ַ Ȯεǰ ־ ͹̿ ߻ ֿ Ÿ ӻ ϰ ִ. ȭ 渮 Ʈε(ָĭ) ϴ.
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ֽż ݴ
  • 2024.03.19 06:59:00 |

    ڳ

    2Ⱓ ֵ ڳ~~~!!!

    0 5 0
ٺ Ϲݾ ǸŰ (2024 05)
౹ 71
ǰ ְ
ѽŻ÷(10) 3,500 2,300 1,200 3,028
޾(100) 25,000 22,000 3,000 23,304
Ʒγΰ(100) 30,000 27,000 3,000 29,237
īɾ(10g) 8,000 5,500 2,500 6,472
Ľõ򿬰(5g) 5,500 4,000 1,500 5,035
Ź(4) 5,000 3,500 1,500 4,449
ڶ(20) 7,000 5,800 1,200 6,433
(10) 6,000 4,000 2,000 4,914
Ժ(10) 4,000 3,000 1,000 3,543
ڱ׸(20) 5,000 3,800 1,200 4,622
ť(10) 3,500 2,300 1,200 2,828
Ȱť(1) 1,200 1,000 200 1,140
Ǯɾ(3.3ml) 25,000 22,000 3,000 24,214
޵𿬰(10g) 7,000 5,000 2,000 6,162
öŸ(34) 13,000 10,000 3,000 12,089
뽺ī(20g) 22,000 18,000 4,000 20,358
ġ(1) 1,100 1,000 100 1,000
ӽ÷(21) 10,000 7,500 2,500 8,998
ͺ(10) 3,500 2,300 1,200 3,138
ݿ(1ڽ) 3,000 2,500 500 2,947
׶÷糪ƮŸ(6) 8,000 7,000 1,000 7,973
߽Ÿ(120) 70,000 40,000 30,000 54,203
Źĸ(10ĸ) 3,000 2,000 1,000 2,941
Ÿ̾(120) 60,000 40,000 20,000 49,168
տ(60ĸ) 30,000 24,000 6,000 27,235
Ÿ̷ER(6) 2,500 2,500 0 2,500
ٿ(30g) 12,000 9,000 3,000 11,221
(120) 25,000 18,000 7,000 21,716
Ʒ(6) 4,000 3,000 1,000 3,509
ǽõĸ(270ĸ) 120,000 85,000 35,000 106,875
B(120) 70,000 60,000 10,000 62,308
׳(10) 3,000 2,000 1,000 2,684
6̺(10) 3,500 2,000 1,500 2,965
(60) 250,000 200,000 50,000 224,000
Ⱦ 12,000 9,000 3,000 10,494
̰źĸ(60ĸ) 25,500 22,000 3,500 23,942
Ųť(20) 5,500 4,500 1,000 4,823
λ絹÷(100) 37,000 29,000 8,000 31,878
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